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7Z21
BAF A12T bound to the lamin A/C Ig-fold domain
9260–9278 Nucleic Acids Research, 2022, Vol. 50, No. 16 Published online 30 August 2022 https://doi.org/10.1093/nar/gkac726 The BAF A12T mutation disrupts lamin A/C interaction, impairing robust repair of nuclear envelope ruptures in Nestor–Guillermo progeria syndrome cells Anne Janssen1, Agathe Marcelot2, Sophia Breus...
7Z22
Connexin43 gap junction channel structure in nanodisc
Qi, Acosta Gutierrez et al. eLife 2023;12:RP87616. DOI: https://doi.org/10.7554/eLife.87616  1 of 27 Structure of the connexin-­43 gap junction channel in a putative closed state Chao Qi1,2†, Silvia Acosta Gutierrez3,4†, Pia Lavriha1,2, Alaa Othman5, Diego Lopez-­Pigozzi6,7, Erva Bayraktar7, Dina Schuster1,2,5, Paol...
7Z23
Connexin43 hemi channel in nanodisc
Qi, Acosta Gutierrez et al. eLife 2023;12:RP87616. DOI: https://doi.org/10.7554/eLife.87616  1 of 27 Structure of the connexin-­43 gap junction channel in a putative closed state Chao Qi1,2†, Silvia Acosta Gutierrez3,4†, Pia Lavriha1,2, Alaa Othman5, Diego Lopez-­Pigozzi6,7, Erva Bayraktar7, Dina Schuster1,2,5, Paol...
7Z24
Cryo-EM structure of HIV-1 reverse transcriptase with a DNA aptamer in complex with nevirapine
Cryo-EM structures of wild-type and E138K/M184I mutant HIV-1 RT/DNA complexed with inhibitors doravirine and rilpivirine Abhimanyu K. Singha,b , Brent De Wijngaerta,b , Marc Bijnensa,b, Kris Uyttersprota,b, Hoai Nguyenc,d , Sergio E. Martineza,b, Dominique Scholsa,b, Piet Herdewijnc,d , Christophe Pannecouquea,b, Eddy ...
7Z26
Crystal structure of YTHDF2 YTH domain in complex with m6A RNA
Fragment Ligands of the m6A‑RNA Reader YTHDF2 Francesco Nai, Raed Nachawati, František Zálešák, Xiang Wang, Yaozong Li,* and Amedeo Caflisch* Cite This: ACS Med. Chem. Lett. 2022, 13, 1500−1509 Read Online ACCESS Metrics & More Article Recommendations * sı Supporting Information ABSTRACT: We report 17 small-molecule ...
7Z27
Crystal structure of the SPOC domain of human RBM15
Article https://doi.org/10.1038/s41467-023-35853-1 The SPOC domain is a phosphoserine binding module that bridges transcription machinery with co- and post-transcriptional regulators Lisa-Marie Appel 1,2,3, Vedran Franke 4, Johannes Benedum 1,2,3,5, Irina Grishkovskaya 6, Xué Strobl3,5, Anton Polyansky 6, Gregor Ammann...
7Z29
Cryo-EM structure of NNRTI resistant M184I/E138K mutant HIV-1 reverse transcriptase with a DNA aptamer in complex with nevirapine
Cryo-EM structures of wild-type and E138K/M184I mutant HIV-1 RT/DNA complexed with inhibitors doravirine and rilpivirine Abhimanyu K. Singha,b , Brent De Wijngaerta,b , Marc Bijnensa,b, Kris Uyttersprota,b, Hoai Nguyenc,d , Sergio E. Martineza,b, Dominique Scholsa,b, Piet Herdewijnc,d , Christophe Pannecouquea,b, Eddy ...
7Z2A
P. berghei kinesin-8B motor domain in no nucleotide state bound to tubulin dimer
Article https://doi.org/10.1038/s41467-022-34710-x Mechanochemical tuning of a kinesin motor essential for malaria parasite transmission Tianyang Liu 1, Fiona Shilliday 1, Alexander D. Cook1,4, Mohammad Zeeshan2, Declan Brady2, Rita Tewari 2, Colin J. Sutherland 3, Anthony J. Roberts 1 & Carolyn A. Moores 1 Plasmodium ...
7Z2B
P. berghei kinesin-8B motor domain in AMPPNP state bound to tubulin dimer
Article https://doi.org/10.1038/s41467-022-34710-x Mechanochemical tuning of a kinesin motor essential for malaria parasite transmission Tianyang Liu 1, Fiona Shilliday 1, Alexander D. Cook1,4, Mohammad Zeeshan2, Declan Brady2, Rita Tewari 2, Colin J. Sutherland 3, Anthony J. Roberts 1 & Carolyn A. Moores 1 Plasmodium ...
7Z2C
P. falciparum kinesin-8B motor domain in no nucleotide bound to tubulin dimer
Article https://doi.org/10.1038/s41467-022-34710-x Mechanochemical tuning of a kinesin motor essential for malaria parasite transmission Tianyang Liu 1, Fiona Shilliday 1, Alexander D. Cook1,4, Mohammad Zeeshan2, Declan Brady2, Rita Tewari 2, Colin J. Sutherland 3, Anthony J. Roberts 1 & Carolyn A. Moores 1 Plasmodium ...
7Z2D
Cryo-EM structure of HIV-1 reverse transcriptase with a DNA aptamer in complex with rilpivirine
Cryo-EM structures of wild-type and E138K/M184I mutant HIV-1 RT/DNA complexed with inhibitors doravirine and rilpivirine Abhimanyu K. Singha,b , Brent De Wijngaerta,b , Marc Bijnensa,b, Kris Uyttersprota,b, Hoai Nguyenc,d , Sergio E. Martineza,b, Dominique Scholsa,b, Piet Herdewijnc,d , Christophe Pannecouquea,b, Eddy ...
7Z2E
Cryo-EM structure of NNRTI resistant M184I/E138K mutant HIV-1 reverse transcriptase with a DNA aptamer in complex with rilpivirine
Cryo-EM structures of wild-type and E138K/M184I mutant HIV-1 RT/DNA complexed with inhibitors doravirine and rilpivirine Abhimanyu K. Singha,b , Brent De Wijngaerta,b , Marc Bijnensa,b, Kris Uyttersprota,b, Hoai Nguyenc,d , Sergio E. Martineza,b, Dominique Scholsa,b, Piet Herdewijnc,d , Christophe Pannecouquea,b, Eddy ...
7Z2G
Cryo-EM structure of HIV-1 reverse transcriptase with a DNA aptamer in complex with doravirine
Cryo-EM structures of wild-type and E138K/M184I mutant HIV-1 RT/DNA complexed with inhibitors doravirine and rilpivirine Abhimanyu K. Singha,b , Brent De Wijngaerta,b , Marc Bijnensa,b, Kris Uyttersprota,b, Hoai Nguyenc,d , Sergio E. Martineza,b, Dominique Scholsa,b, Piet Herdewijnc,d , Christophe Pannecouquea,b, Eddy ...
7Z2H
Cryo-EM structure of NNRTI resistant M184I/E138K mutant HIV-1 reverse transcriptase with a DNA aptamer in complex with doravirine
Cryo-EM structures of wild-type and E138K/M184I mutant HIV-1 RT/DNA complexed with inhibitors doravirine and rilpivirine Abhimanyu K. Singha,b , Brent De Wijngaerta,b , Marc Bijnensa,b, Kris Uyttersprota,b, Hoai Nguyenc,d , Sergio E. Martineza,b, Dominique Scholsa,b, Piet Herdewijnc,d , Christophe Pannecouquea,b, Eddy ...
7Z2J
White Bream virus N7-Methyltransferase
11186–11198 Nucleic Acids Research, 2022, Vol. 50, No. 19 Published online 21 October 2022 https://doi.org/10.1093/nar/gkac876 A second type of N7-guanine RNA cap methyltransferase in an unusual locus of a large RNA virus genome Ashleigh Shannon 1,†, Bhawna Sama 1,†, Pierre Gauffre 1, Th´eo Guez2, Franc¸oise Debart 2, ...
7Z2K
Crystal structure of SARS-CoV-2 Main Protease in orthorhombic space group p212121
Article https://doi.org/10.1038/s41467-024-48109-3 SARS-CoV-2 Mpro responds to oxidation by forming disulfide and NOS/SONOS bonds A list of authors and their affiliations appears at the end of the paper The main protease (Mpro) of SARS-CoV-2 is critical for viral function and a key drug target. Mpro is only active when r...
7Z2M
Crystal Structure of the 11.003 Fab in complex with human IL-17A
ARTICLE “Redirecting an anti-IL-1β antibody to bind a new, unrelated and computationally predicted epitope on hIL-17A” Sharon Fischman1,8, Itay Levin1,4,8, Jean-Michel Rondeau 2, Marek Štrajbl 1, Sylvie Lehmann2, Thomas Huber2,5, Guy Nimrod 1✉, Régis Cebe2, Dotan Omer1,6, Jiri Kovarik2, Shmuel Bernstein1, Yehezkel Sass...
7Z2O
PARP15 catalytic domain in complex with OUL215
[1,2,4]Triazolo[3,4‑b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes Sudarshan Murthy,⊥Maria Giulia Nizi,⊥Mirko M. Maksimainen,⊥Serena Massari, Juho Alaviuhkola, Barbara E. Lippok, Chiara Vagaggini, Sven T. Sowa, Albert Galera-Prat, Yashwanth Ashok, Harika...
7Z2Q
PARP15 catalytic domain in complex with OUL232
[1,2,4]Triazolo[3,4‑b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes Sudarshan Murthy,⊥Maria Giulia Nizi,⊥Mirko M. Maksimainen,⊥Serena Massari, Juho Alaviuhkola, Barbara E. Lippok, Chiara Vagaggini, Sven T. Sowa, Albert Galera-Prat, Yashwanth Ashok, Harika...
7Z2S
Escherichia coli periplasmic phytase AppA, complex with myo-inositol hexakissulfate
Citation: Acquistapace, I.M.; Thompson, E.J.; Kühn, I.; Bedford, M.R.; Brearley, C.A.; Hemmings, A.M. Insights to the Structural Basis for the Stereospecificity of the Escherichia coli Phytase, AppA. Int. J. Mol. Sci. 2022, 23, 6346. https://doi.org/10.3390/ ijms23116346 Academic Editors: Antonio Zuorro, Yung-Chuan Liu ...
7Z2T
Escherichia coli periplasmic phytase AppA D304A mutant, complex with myo-inositol hexakissulfate
Citation: Acquistapace, I.M.; Thompson, E.J.; Kühn, I.; Bedford, M.R.; Brearley, C.A.; Hemmings, A.M. Insights to the Structural Basis for the Stereospecificity of the Escherichia coli Phytase, AppA. Int. J. Mol. Sci. 2022, 23, 6346. https://doi.org/10.3390/ ijms23116346 Academic Editors: Antonio Zuorro, Yung-Chuan Liu ...
7Z2U
Wild-type ferulic acid esterase from Lactobacillus buchneri in complex with ferulate
Frontiers in Microbiology 01 frontiersin.org Crystal structure of the feruloyl esterase from Lentilactobacillus buchneri reveals a novel homodimeric state Kamyar Mogodiniyai Kasmaei 1,2, Dayanand C. Kalyani 1, Tom Reichenbach 1, Amparo Jiménez-Quero 3, Francisco Vilaplana 3 and Christina Divne 1* 1 Department of I...
7Z2V
Ferulic acid esterase variant S114A from Lactobacillus buchneri
Frontiers in Microbiology 01 frontiersin.org Crystal structure of the feruloyl esterase from Lentilactobacillus buchneri reveals a novel homodimeric state Kamyar Mogodiniyai Kasmaei 1,2, Dayanand C. Kalyani 1, Tom Reichenbach 1, Amparo Jiménez-Quero 3, Francisco Vilaplana 3 and Christina Divne 1* 1 Department of I...
7Z2W
Escherichia coli periplasmic phytase AppA D304A,T305E mutant, complex with myo-inositol hexakissulfate
Citation: Acquistapace, I.M.; Thompson, E.J.; Kühn, I.; Bedford, M.R.; Brearley, C.A.; Hemmings, A.M. Insights to the Structural Basis for the Stereospecificity of the Escherichia coli Phytase, AppA. Int. J. Mol. Sci. 2022, 23, 6346. https://doi.org/10.3390/ ijms23116346 Academic Editors: Antonio Zuorro, Yung-Chuan Liu ...
7Z2X
Wild-type ferulic acid esterase from Lactobacillus buchneri
Frontiers in Microbiology 01 frontiersin.org Crystal structure of the feruloyl esterase from Lentilactobacillus buchneri reveals a novel homodimeric state Kamyar Mogodiniyai Kasmaei 1,2, Dayanand C. Kalyani 1, Tom Reichenbach 1, Amparo Jiménez-Quero 3, Francisco Vilaplana 3 and Christina Divne 1* 1 Department of I...
7Z2Y
Escherichia coli periplasmic phytase AppA T305E mutant, complex with myo-inositol hexakissulfate
Citation: Acquistapace, I.M.; Thompson, E.J.; Kühn, I.; Bedford, M.R.; Brearley, C.A.; Hemmings, A.M. Insights to the Structural Basis for the Stereospecificity of the Escherichia coli Phytase, AppA. Int. J. Mol. Sci. 2022, 23, 6346. https://doi.org/10.3390/ ijms23116346 Academic Editors: Antonio Zuorro, Yung-Chuan Liu ...
7Z2Z
Structure of yeast RNA Polymerase III-DNA-Ty1 integrase complex (Pol III-DNA-IN1) at 3.1 A
Article https://doi.org/10.1038/s41467-023-37109-4 Structural basis of Ty1 integrase tethering to RNA polymerase III for targeted retrotransposon integration Phong Quoc Nguyen 1,2,6, Sonia Huecas1,6, Amna Asif-Laidin 3,6, Adrián Plaza-Pegueroles 1, Beatrice Capuzzi3, Noé Palmic3, Christine Conesa4, Joël Acker 4, Juan R...
7Z30
Structure of yeast RNA Polymerase III-Ty1 integrase complex at 2.9 A (focus subunit C11 terminal Zn-ribbon in the funnel pore).
Article https://doi.org/10.1038/s41467-023-37109-4 Structural basis of Ty1 integrase tethering to RNA polymerase III for targeted retrotransposon integration Phong Quoc Nguyen 1,2,6, Sonia Huecas1,6, Amna Asif-Laidin 3,6, Adrián Plaza-Pegueroles 1, Beatrice Capuzzi3, Noé Palmic3, Christine Conesa4, Joël Acker 4, Juan R...
7Z31
Structure of yeast RNA Polymerase III-Ty1 integrase complex at 2.7 A (focus subunit C11, no C11 C-terminal Zn-ribbon in the funnel pore).
Article https://doi.org/10.1038/s41467-023-37109-4 Structural basis of Ty1 integrase tethering to RNA polymerase III for targeted retrotransposon integration Phong Quoc Nguyen 1,2,6, Sonia Huecas1,6, Amna Asif-Laidin 3,6, Adrián Plaza-Pegueroles 1, Beatrice Capuzzi3, Noé Palmic3, Christine Conesa4, Joël Acker 4, Juan R...
7Z32
Escherichia coli periplasmic phytase AppA D304A mutant, phosphohistidine intermediate
Citation: Acquistapace, I.M.; Thompson, E.J.; Kühn, I.; Bedford, M.R.; Brearley, C.A.; Hemmings, A.M. Insights to the Structural Basis for the Stereospecificity of the Escherichia coli Phytase, AppA. Int. J. Mol. Sci. 2022, 23, 6346. https://doi.org/10.3390/ ijms23116346 Academic Editors: Antonio Zuorro, Yung-Chuan Liu ...
7Z34
Structure of pre-60S particle bound to DRG1(AFG2).
Articles https://doi.org/10.1038/s41594-022-00832-5 1Institute of Molecular Biosciences, University of Graz, Graz, Austria. 2BioTechMed-Graz, Graz, Austria. 3Research Institute of Molecular Pathology (IMP), Vienna BioCenter, Vienna, Austria. 4Institute of Science and Technology Austria, Klosterneuburg, Austria. 5Depar...
7Z36
Crystal structure of the KAP1 tripartite motif in complex with the ZNF93 KRAB domain
Article Structure and functional mapping of the KRAB-KAP1 repressor complex Guido A Stoll1,2 , Ninoslav Pandiloski3 , Christopher H Douse3 & Yorgo Modis1,2,* Abstract Transposable elements are a genetic reservoir from which new genes and regulatory elements can emerge. However, expression of transposable elements can b...
7Z39
Structure of Belumosudil bound to CK2alpha
research communications 348 https://doi.org/10.1107/S2053230X22008767 Acta Cryst. (2022). F78, 348–353 Received 24 June 2022 Accepted 1 September 2022 Edited by S. Sheriff, Bristol-Myers Squibb, USA Keywords: belumosudil; CK2 inhibition; Rho-associated coiled-coil kinase 2; ROCK2 inhibition; kinase inhibitors; selecti...
7Z3A
AMC009 SOSIPv5.2 in complex with Fabs ACS101 and ACS124
nature communications Article https://doi.org/10.1038/s41467-022-32208-0 Identification of IOMA-class neutralizing antibodies targeting the CD4-binding site on the HIV-1 envelope glycoprotein Jelle van Schooten 1, Elinaz Farokhi 2, Anna Schorcht1, Tom L. G. M. van den Kerkhof1, Hongmei Gao3, Patricia van der Woude1, Jud...
7Z3C
Solution structure of GltJ GYF domain from Myxococcus xanthus
Attia et al., Sci. Adv. 10, eadn2789 (2024) 29 May 2024 S c i e n c e A d va n c e s | R e s e a r c h A r t i c l e 1 of 15 M I C R O B I O LO G Y A molecular switch controls assembly of bacterial focal adhesions Bouchra Attia1†, Laetitia My2†, Jean Philippe Castaing2, Céline Dinet2, Hugo Le Guenno3, Victori...
7Z3D
XFEL structure of Class Ib ribonucleotide reductase dimanganese(II) NrdF in complex with oxidized NrdI from Bacillus cereus
John et al. eLife 2022;11:e79226. DOI: https://doi.org/10.7554/eLife.79226  1 of 23 Redox-­controlled reorganization and flavin strain within the ribonucleotide reductase R2b–NrdI complex monitored by serial femtosecond crystallography Juliane John1, Oskar Aurelius1,2, Vivek Srinivas1, Patricia Saura1, In-­Sik Kim3...
7Z3E
XFEL structure of Class Ib ribonucleotide reductase dimanganese(II) NrdF in complex with hydroquinone NrdI from Bacillus cereus
John et al. eLife 2022;11:e79226. DOI: https://doi.org/10.7554/eLife.79226  1 of 23 Redox-­controlled reorganization and flavin strain within the ribonucleotide reductase R2b–NrdI complex monitored by serial femtosecond crystallography Juliane John1, Oskar Aurelius1,2, Vivek Srinivas1, Patricia Saura1, In-­Sik Kim3...
7Z3H
Crystal structure of Iba57 from Chaetomium thermophilum
The iron–sulfur cluster assembly (ISC) protein Iba57 executes a tetrahydrofolate-independent function in mitochondrial [4Fe–4S] protein maturation Received for publication, June 3, 2022, and in revised form, August 23, 2022 Published, Papers in Press, September 6, 2022, https://doi.org/10.1016/j.jbc.2022.102465 Ulrich ...
7Z3J
Structure of crystallisable rat Phospholipase C gamma 1 in complex with inositol 1,4,5-trisphosphate
Le Huray et al., Sci. Adv. 8, eabp9688 (2022) 24 June 2022 SCIE N C E A D V A NCES | RESEA R CH A RT ICL E 1 of 15 BI O PH YSICS Characterization of the membrane interactions of phospholipase C reveals key features of the  active enzyme Kyle I. P. Le Huray1,2,3, Tom D. Bunney4*, Nikos Pinotsis5, Antreas C. Kall...
7Z3N
Cryo-EM structure of the ribosome-associated RAC complex on the 80S ribosome - RAC-1 conformation
Nature Structural & Molecular Biology | Volume 30 | May 2023 | 670–677 670 nature structural & molecular biology Article https://doi.org/10.1038/s41594-023-00973-1 Structural inventory of cotranslational protein folding by the eukaryotic RAC complex Miglė Kišonaitė    , Klemens Wild    , Karine Lapouge, Genís Valentí...
7Z3O
Cryo-EM structure of the ribosome-associated RAC complex on the 80S ribosome - RAC-2 conformation
Nature Structural & Molecular Biology | Volume 30 | May 2023 | 670–677 670 nature structural & molecular biology Article https://doi.org/10.1038/s41594-023-00973-1 Structural inventory of cotranslational protein folding by the eukaryotic RAC complex Miglė Kišonaitė    , Klemens Wild    , Karine Lapouge, Genís Valentí...
7Z3T
Crystal structure of apo human Cathepsin L
ARTICLE Calpeptin is a potent cathepsin inhibitor and drug candidate for SARS-CoV-2 infections Patrick Y. A. Reinke 1,22, Edmarcia Elisa de Souza2,22, Sebastian Günther 1,22, Sven Falke 1, Julia Lieske 1, Wiebke Ewert 1, Jure Loboda 3,4, Alexander Herrmann 5, Aida Rahmani Mashhour 1, Katarina Karničar 3,6, Aleksandra U...
7Z3U
Crystal structure of SARS-CoV-2 Main Protease after incubation with Sulfo-Calpeptin
ARTICLE Calpeptin is a potent cathepsin inhibitor and drug candidate for SARS-CoV-2 infections Patrick Y. A. Reinke 1,22, Edmarcia Elisa de Souza2,22, Sebastian Günther 1,22, Sven Falke 1, Julia Lieske 1, Wiebke Ewert 1, Jure Loboda 3,4, Alexander Herrmann 5, Aida Rahmani Mashhour 1, Katarina Karničar 3,6, Aleksandra U...
7Z3V
Escherichia coli periplasmic phytase AppA D304E mutant, complex with myo-inositol hexakissulfate
Citation: Acquistapace, I.M.; Thompson, E.J.; Kühn, I.; Bedford, M.R.; Brearley, C.A.; Hemmings, A.M. Insights to the Structural Basis for the Stereospecificity of the Escherichia coli Phytase, AppA. Int. J. Mol. Sci. 2022, 23, 6346. https://doi.org/10.3390/ ijms23116346 Academic Editors: Antonio Zuorro, Yung-Chuan Liu ...
7Z3W
Crystal structure of the AAL160 Fab
ARTICLE “Redirecting an anti-IL-1β antibody to bind a new, unrelated and computationally predicted epitope on hIL-17A” Sharon Fischman1,8, Itay Levin1,4,8, Jean-Michel Rondeau 2, Marek Štrajbl 1, Sylvie Lehmann2, Thomas Huber2,5, Guy Nimrod 1✉, Régis Cebe2, Dotan Omer1,6, Jiri Kovarik2, Shmuel Bernstein1, Yehezkel Sass...
7Z3Y
Structure of the mouse 8-oxoguanine DNA Glycosylase mOGG1 in complex with ligand TH013545
Article https://doi.org/10.1038/s41467-025-56893-9 Virtual fragment screening for DNA repair inhibitors in vast chemical space Andreas Luttens 1,2,3, Duc Duy Vo1, Emma R. Scaletti4, Elisée Wiita5, Ingrid Almlöf5, Olov Wallner5, Jonathan Davies4, Sara Košenina 4, Liuzhen Meng5, Maeve Long5, Oliver Mortusewicz 5, Geoffre...
7Z41
PARP15 catalytic domain in complex with OUL209
[1,2,4]Triazolo[3,4‑b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes Sudarshan Murthy,⊥Maria Giulia Nizi,⊥Mirko M. Maksimainen,⊥Serena Massari, Juho Alaviuhkola, Barbara E. Lippok, Chiara Vagaggini, Sven T. Sowa, Albert Galera-Prat, Yashwanth Ashok, Harika...
7Z42
Influenza B polymerase with Pol II pSer5 CTD peptide mimic bound in site 2B
RESEARCH ARTICLE Type B and type A influenza polymerases have evolved distinct binding interfaces to recruit the RNA polymerase II CTD Tim Krischuns1, Catherine Isel1, Petra Drncova2, Maria Lukarska2¤, Alexander Pflug2, Sylvain Paisant1, Vincent Navratil3, Stephen CusackID2*, Nadia NaffakhID1* 1 Institut Pasteur, Unive...
7Z43
Influenza B polymerase with Pol II pSer5 CTD peptide mimic bound in site 1B and 2B
RESEARCH ARTICLE Type B and type A influenza polymerases have evolved distinct binding interfaces to recruit the RNA polymerase II CTD Tim Krischuns1, Catherine Isel1, Petra Drncova2, Maria Lukarska2¤, Alexander Pflug2, Sylvain Paisant1, Vincent Navratil3, Stephen CusackID2*, Nadia NaffakhID1* 1 Institut Pasteur, Unive...
7Z44
Portal of bacteriophage SU10
Article https://doi.org/10.1038/s41467-022-33305-w Tail proteins of phage SU10 reorganize into the nozzle for genome delivery Marta Šiborová 1, Tibor Füzik 1, Michaela Procházková 1, Jiří Nováček1, Martin Benešík2, Anders S. Nilsson 3 & Pavel Plevka 1 Escherichia coli phage SU10 belongs to the genus Kuravirus from the ...
7Z45
Central part (C10) of bacteriophage SU10 capsid
Article https://doi.org/10.1038/s41467-022-33305-w Tail proteins of phage SU10 reorganize into the nozzle for genome delivery Marta Šiborová 1, Tibor Füzik 1, Michaela Procházková 1, Jiří Nováček1, Martin Benešík2, Anders S. Nilsson 3 & Pavel Plevka 1 Escherichia coli phage SU10 belongs to the genus Kuravirus from the ...
7Z46
Top part (C5) of bacteriophage SU10 capsid
Article https://doi.org/10.1038/s41467-022-33305-w Tail proteins of phage SU10 reorganize into the nozzle for genome delivery Marta Šiborová 1, Tibor Füzik 1, Michaela Procházková 1, Jiří Nováček1, Martin Benešík2, Anders S. Nilsson 3 & Pavel Plevka 1 Escherichia coli phage SU10 belongs to the genus Kuravirus from the ...
7Z47
Tail of bacteriophage SU10
Article https://doi.org/10.1038/s41467-022-33305-w Tail proteins of phage SU10 reorganize into the nozzle for genome delivery Marta Šiborová 1, Tibor Füzik 1, Michaela Procházková 1, Jiří Nováček1, Martin Benešík2, Anders S. Nilsson 3 & Pavel Plevka 1 Escherichia coli phage SU10 belongs to the genus Kuravirus from the ...
7Z48
Bottom part (C5) of bacteriophage SU10 capsid
Article https://doi.org/10.1038/s41467-022-33305-w Tail proteins of phage SU10 reorganize into the nozzle for genome delivery Marta Šiborová 1, Tibor Füzik 1, Michaela Procházková 1, Jiří Nováček1, Martin Benešík2, Anders S. Nilsson 3 & Pavel Plevka 1 Escherichia coli phage SU10 belongs to the genus Kuravirus from the ...
7Z49
The capsid of bacteriophage SU10.
Article https://doi.org/10.1038/s41467-022-33305-w Tail proteins of phage SU10 reorganize into the nozzle for genome delivery Marta Šiborová 1, Tibor Füzik 1, Michaela Procházková 1, Jiří Nováček1, Martin Benešík2, Anders S. Nilsson 3 & Pavel Plevka 1 Escherichia coli phage SU10 belongs to the genus Kuravirus from the ...
7Z4A
Bacteriophage SU10 tail and bottom part of the capsid (C1)
Article https://doi.org/10.1038/s41467-022-33305-w Tail proteins of phage SU10 reorganize into the nozzle for genome delivery Marta Šiborová 1, Tibor Füzik 1, Michaela Procházková 1, Jiří Nováček1, Martin Benešík2, Anders S. Nilsson 3 & Pavel Plevka 1 Escherichia coli phage SU10 belongs to the genus Kuravirus from the ...
7Z4B
Bacteriophage SU10 virion (C1)
Article https://doi.org/10.1038/s41467-022-33305-w Tail proteins of phage SU10 reorganize into the nozzle for genome delivery Marta Šiborová 1, Tibor Füzik 1, Michaela Procházková 1, Jiří Nováček1, Martin Benešík2, Anders S. Nilsson 3 & Pavel Plevka 1 Escherichia coli phage SU10 belongs to the genus Kuravirus from the ...
7Z4C
SpCas9 bound to 6 nucleotide complementary DNA substrate
Nature  |  Vol 609  |  1 September 2022  |  191 Article R-loop formation and conformational activation mechanisms of Cas9 Martin Pacesa1, Luuk Loeff1,2, Irma Querques1,2, Lena M. Muckenfuss1,2, Marta Sawicka1 & Martin Jinek1 ✉ Cas9 is a CRISPR-associated endonuclease capable of RNA-guided, site-specific DNA cleavage...
7Z4D
Crystal structure of SpCas9 bound to a 10 nucleotide complementary DNA substrate
Nature  |  Vol 609  |  1 September 2022  |  191 Article R-loop formation and conformational activation mechanisms of Cas9 Martin Pacesa1, Luuk Loeff1,2, Irma Querques1,2, Lena M. Muckenfuss1,2, Marta Sawicka1 & Martin Jinek1 ✉ Cas9 is a CRISPR-associated endonuclease capable of RNA-guided, site-specific DNA cleavage...
7Z4E
SpCas9 bound to 8-nucleotide complementary DNA substrate
Nature  |  Vol 609  |  1 September 2022  |  191 Article R-loop formation and conformational activation mechanisms of Cas9 Martin Pacesa1, Luuk Loeff1,2, Irma Querques1,2, Lena M. Muckenfuss1,2, Marta Sawicka1 & Martin Jinek1 ✉ Cas9 is a CRISPR-associated endonuclease capable of RNA-guided, site-specific DNA cleavage...
7Z4F
Tail of phage SU10 genome release intermediate
Article https://doi.org/10.1038/s41467-022-33305-w Tail proteins of phage SU10 reorganize into the nozzle for genome delivery Marta Šiborová 1, Tibor Füzik 1, Michaela Procházková 1, Jiří Nováček1, Martin Benešík2, Anders S. Nilsson 3 & Pavel Plevka 1 Escherichia coli phage SU10 belongs to the genus Kuravirus from the ...
7Z4G
SpCas9 bound to 12-nucleotide complementary DNA substrate
Nature  |  Vol 609  |  1 September 2022  |  191 Article R-loop formation and conformational activation mechanisms of Cas9 Martin Pacesa1, Luuk Loeff1,2, Irma Querques1,2, Lena M. Muckenfuss1,2, Marta Sawicka1 & Martin Jinek1 ✉ Cas9 is a CRISPR-associated endonuclease capable of RNA-guided, site-specific DNA cleavage...
7Z4H
SpCas9 bound to 14-nucleotide complementary DNA substrate
Nature  |  Vol 609  |  1 September 2022  |  191 Article R-loop formation and conformational activation mechanisms of Cas9 Martin Pacesa1, Luuk Loeff1,2, Irma Querques1,2, Lena M. Muckenfuss1,2, Marta Sawicka1 & Martin Jinek1 ✉ Cas9 is a CRISPR-associated endonuclease capable of RNA-guided, site-specific DNA cleavage...
7Z4I
SpCas9 bound to 16-nucleotide complementary DNA substrate
Nature  |  Vol 609  |  1 September 2022  |  191 Article R-loop formation and conformational activation mechanisms of Cas9 Martin Pacesa1, Luuk Loeff1,2, Irma Querques1,2, Lena M. Muckenfuss1,2, Marta Sawicka1 & Martin Jinek1 ✉ Cas9 is a CRISPR-associated endonuclease capable of RNA-guided, site-specific DNA cleavage...
7Z4J
SpCas9 bound to 18-nucleotide complementary DNA substrate in the catalytic state
Nature  |  Vol 609  |  1 September 2022  |  191 Article R-loop formation and conformational activation mechanisms of Cas9 Martin Pacesa1, Luuk Loeff1,2, Irma Querques1,2, Lena M. Muckenfuss1,2, Marta Sawicka1 & Martin Jinek1 ✉ Cas9 is a CRISPR-associated endonuclease capable of RNA-guided, site-specific DNA cleavage...
7Z4K
SpCas9 bound to 10-nucleotide complementary DNA substrate
Nature  |  Vol 609  |  1 September 2022  |  191 Article R-loop formation and conformational activation mechanisms of Cas9 Martin Pacesa1, Luuk Loeff1,2, Irma Querques1,2, Lena M. Muckenfuss1,2, Marta Sawicka1 & Martin Jinek1 ✉ Cas9 is a CRISPR-associated endonuclease capable of RNA-guided, site-specific DNA cleavage...
7Z4L
SpCas9 bound to 18-nucleotide complementary DNA substrate in the checkpoint state
Nature  |  Vol 609  |  1 September 2022  |  191 Article R-loop formation and conformational activation mechanisms of Cas9 Martin Pacesa1, Luuk Loeff1,2, Irma Querques1,2, Lena M. Muckenfuss1,2, Marta Sawicka1 & Martin Jinek1 ✉ Cas9 is a CRISPR-associated endonuclease capable of RNA-guided, site-specific DNA cleavage...
7Z4O
Influenza A/H7N9 polymerase core dimer with Pol II pSer5 CTD peptide mimic bound in site 2A
RESEARCH ARTICLE Type B and type A influenza polymerases have evolved distinct binding interfaces to recruit the RNA polymerase II CTD Tim Krischuns1, Catherine Isel1, Petra Drncova2, Maria Lukarska2¤, Alexander Pflug2, Sylvain Paisant1, Vincent Navratil3, Stephen CusackID2*, Nadia NaffakhID1* 1 Institut Pasteur, Unive...
7Z4S
Crystal structure of SARS-CoV-2 Mpro in complex with cyclic peptide GM4 including unnatural amino acids.
Nature Chemistry | Volume 15 | July 2023 | 998–1005 998 nature chemistry Article https://doi.org/10.1038/s41557-023-01205-1 In vitro selection of macrocyclic peptide inhibitors containing cyclic γ2,4-amino acids targeting the SARS-CoV-2 main protease Takashi Miura    1, Tika R. Malla    2, C. David Owen3,4, Anthony T...
7Z4T
AAL160 FAB IN COMPLEX WITH HUMAN INTERLEUKIN-1 BETA
ARTICLE “Redirecting an anti-IL-1β antibody to bind a new, unrelated and computationally predicted epitope on hIL-17A” Sharon Fischman1,8, Itay Levin1,4,8, Jean-Michel Rondeau 2, Marek Štrajbl 1, Sylvie Lehmann2, Thomas Huber2,5, Guy Nimrod 1✉, Régis Cebe2, Dotan Omer1,6, Jiri Kovarik2, Shmuel Bernstein1, Yehezkel Sass...
7Z4U
Crystal structure of YTHDF2 with compound YLI_DF_028
Fragment Ligands of the m6A‑RNA Reader YTHDF2 Francesco Nai, Raed Nachawati, František Zálešák, Xiang Wang, Yaozong Li,* and Amedeo Caflisch* Cite This: ACS Med. Chem. Lett. 2022, 13, 1500−1509 Read Online ACCESS Metrics & More Article Recommendations * sı Supporting Information ABSTRACT: We report 17 small-molecule ...
7Z4W
gp6/gp15/gp16 connector complex of bacteriophage SPP1
Article https://doi.org/10.1038/s41467-022-34999-8 CryoEM structure and assembly mechanism of a bacterial virus genome gatekeeper Igor Orlov1,5,6, Stéphane Roche2,6, Sandrine Brasilès2, Natalya Lukoyanova 3, Marie-Christine Vaney4, Paulo Tavares 2 & Elena V. Orlova 3 Numerous viruses package their dsDNA genome into pre...
7Z50
Structure of the highly diabetogenic 4.1-T cell receptor targeting a hybrid insulin peptide bound to I-Ag7.
Structural plasticity in I-Ag7 links autoreactivity to hybrid insulin peptides in type I diabetes Elena Erausquin 1,2,3†, Pau Serra 4†, Daniel Parras 4†, Pere Santamaria 4,5* and Jacinto Lo´ pez-Sagaseta 1,2,3*‡ 1Unit of Protein Crystallography and Structural Immunology, Navarrabiomed, Navarra, Spain, 2Public Universit...
7Z51
Tick-borne encephalitis virus Kuutsalo-14
  Citation: Pulkkinen, L.I.A.; Barrass, S.V.; Domanska, A.; Överby, A.K.; Anastasina, M.; Butcher, S.J. Molecular Organisation of Tick-Borne Encephalitis Virus. Viruses 2022, 14, 792. https://doi.org/10.3390/ v14040792 Academic Editors: David Stuart and Elizabeth Fry Received: 25 March 2022 Accepted: 7 ...
7Z53
Structure of native leukocyte myeloperoxidase in complex with a truncated version (SPIN truncated) of the Staphyloccal Peroxidase Inhibitor SPIN from Staphylococcus aureus
The staphylococcal inhibitory protein SPIN binds to human myeloperoxidase with picomolar affinity but only dampens halide oxidation Received for publication, July 13, 2022, and in revised form, September 15, 2022 Published, Papers in Press, September 21, 2022, https://doi.org/10.1016/j.jbc.2022.102514 Urban Leitgeb1, Pa...
7Z54
Crystal structure of YTHDF2 with compound YLI_DC1_006
Fragment Ligands of the m6A‑RNA Reader YTHDF2 Francesco Nai, Raed Nachawati, František Zálešák, Xiang Wang, Yaozong Li,* and Amedeo Caflisch* Cite This: ACS Med. Chem. Lett. 2022, 13, 1500−1509 Read Online ACCESS Metrics & More Article Recommendations * sı Supporting Information ABSTRACT: We report 17 small-molecule ...
7Z55
Crystal Structure of the Ring Nuclease 0455 from Sulfolobus islandicus (Sis0455) in complex with its substrate
Published online 22 October 2022 Nucleic Acids Research, 2022, Vol. 50, No. 19 11199–11213 https://doi.org/10.1093/nar/gkac923 Molecular basis of cyclic tetra-oligoadenylate processing by small standalone CRISPR-Cas ring nucleases Rafael Molina 1,*, Ricardo Garcia-Martin 1, Blanca L´opez-M´endez2, Anne Louise Grøn Jens...
7Z56
Crystal Structure of the Ring Nuclease 0455 from Sulfolobus islandicus (Sis0455) in its apo form
Published online 22 October 2022 Nucleic Acids Research, 2022, Vol. 50, No. 19 11199–11213 https://doi.org/10.1093/nar/gkac923 Molecular basis of cyclic tetra-oligoadenylate processing by small standalone CRISPR-Cas ring nucleases Rafael Molina 1,*, Ricardo Garcia-Martin 1, Blanca L´opez-M´endez2, Anne Louise Grøn Jens...
7Z57
Crystal structure of Human Serum Albumin in complex with surfactant GenX (2,3,3,3-tetrafluoro-2-(heptafluoropropoxy) propanoate)
Investigation of the Interaction between Human Serum Albumin and Branched Short-Chain Perfluoroalkyl Compounds Giulia Moro, Stefano Liberi, Filippo Vascon, Sara Linciano, Sofia De Felice, Silvano Fasolato, Carlo Foresta, Luca De Toni, Andrea Di Nisio, Laura Cendron,* and Alessandro Angelini* Cite This: Chem. Res. Toxic...
7Z58
Crystal structure of human Cathepsin L in complex with covalently bound Calpeptin
ARTICLE Calpeptin is a potent cathepsin inhibitor and drug candidate for SARS-CoV-2 infections Patrick Y. A. Reinke 1,22, Edmarcia Elisa de Souza2,22, Sebastian Günther 1,22, Sven Falke 1, Julia Lieske 1, Wiebke Ewert 1, Jure Loboda 3,4, Alexander Herrmann 5, Aida Rahmani Mashhour 1, Katarina Karničar 3,6, Aleksandra U...
7Z59
SARS-CoV-2 main protease (Mpro) covalently modified with a penicillin derivative
Penicillin Derivatives Inhibit the SARS-CoV‑2 Main Protease by Reaction with Its Nucleophilic Cysteine Tika R. Malla,∥Lennart Brewitz,*,∥Dorian-Gabriel Muntean, Hiba Aslam, C. David Owen, Eidarus Salah, Anthony Tumber, Petra Lukacik, Claire Strain-Damerell, Halina Mikolajek, Martin A. Walsh, and Christopher J. Schofield...
7Z5A
Crystal structure of the trapped complex of mouse Endonuclease VIII-LIKE 3 (mNEIL3) and hairpin DNA with 5'overhang
10436–10448 Nucleic Acids Research, 2022, Vol. 50, No. 18 Published online 26 September 2022 https://doi.org/10.1093/nar/gkac793 Model of abasic site DNA cross-link repair; from the architecture of NEIL3 DNA binding domains to the X-structure model Andrea Huskova1, Dhurvas Chandrasekaran Dinesh 1, Pavel Srb1, Evzen Bou...
7Z5B
Structure of the mouse 8-oxoguanine DNA Glycosylase mOGG1 in complex with ligand TH013546
Article https://doi.org/10.1038/s41467-025-56893-9 Virtual fragment screening for DNA repair inhibitors in vast chemical space Andreas Luttens 1,2,3, Duc Duy Vo1, Emma R. Scaletti4, Elisée Wiita5, Ingrid Almlöf5, Olov Wallner5, Jonathan Davies4, Sara Košenina 4, Liuzhen Meng5, Maeve Long5, Oliver Mortusewicz 5, Geoffre...
7Z5C
Chimera of AP2 with FCHO2 linker domain as a fusion on Cmu2 subunit
Zaccai et al., Sci. Adv. 8, eabn2018 (2022) 29 April 2022 SCIE N C E A D V A NCES | RESEA R CH A RT ICL E 1 of 21 ST RUCTURAL B IOL OG Y FCHO controls AP2’s initiating role in endocytosis through a PtdIns(4,5)P2-dependent switch Nathan R. Zaccai1†, Zuzana Kadlecova1*†, Veronica Kane Dickson1, Kseniya Korobchevska...
7Z5I
Transcription factor MYF5 bound to symmetrical site
Nature Structural & Molecular Biology | Volume 32 | April 2025 | 650–661 650 nature structural & molecular biology Article https://doi.org/10.1038/s41594-024-01449-6 Interfacial water confers transcription factors with dinucleotide specificity Ekaterina Morgunova    1, Gabor Nagy    2, Yimeng Yin    3,4, Fangjie Zhu  ...
7Z5K
Transcription factor MYF5 bound to non-symmetrical site
Nature Structural & Molecular Biology | Volume 32 | April 2025 | 650–661 650 nature structural & molecular biology Article https://doi.org/10.1038/s41594-024-01449-6 Interfacial water confers transcription factors with dinucleotide specificity Ekaterina Morgunova    1, Gabor Nagy    2, Yimeng Yin    3,4, Fangjie Zhu  ...
7Z5M
Crystal structure of YTHDF2 with compound YLI_DC1_008
Fragment Ligands of the m6A‑RNA Reader YTHDF2 Francesco Nai, Raed Nachawati, František Zálešák, Xiang Wang, Yaozong Li,* and Amedeo Caflisch* Cite This: ACS Med. Chem. Lett. 2022, 13, 1500−1509 Read Online ACCESS Metrics & More Article Recommendations * sı Supporting Information ABSTRACT: We report 17 small-molecule ...
7Z5O
W-formate dehydrogenase from Desulfovibrio vulgaris - Dithionite reduced form
Spectroscopic and Structural Characterization of Reduced Desulfovibrio vulgaris Hildenborough W‑FdhAB Reveals Stable Metal Coordination during Catalysis Ana Rita Oliveira, Cristiano Mota, Kateryna Klymanska, Frédéric Biaso, Maria João Romão,* Bruno Guigliarelli,* and Inês Cardoso Pereira* Cite This: ACS Chem. Biol. ...
7Z5P
Bilirubin oxidase from Bacillus pumilus
Citation: Gihaz, S.; Herzallh, N.S.; Cohen, Y.; Bachar, O.; Fishman, A.; Yehezkeli, O. The Structure of Bilirubin Oxidase from Bacillus pumilus Reveals a Unique Disulfide Bond for Site-Specific Direct Electron Transfer. Biosensors 2022, 12, 258. https://doi.org/10.3390/ bios12050258 Received: 14 March 2022 Accepted: 15 A...
7Z5R
Structure of the mouse 8-oxoguanine DNA Glycosylase mOGG1 in complex with ligand TH012035
Article https://doi.org/10.1038/s41467-025-56893-9 Virtual fragment screening for DNA repair inhibitors in vast chemical space Andreas Luttens 1,2,3, Duc Duy Vo1, Emma R. Scaletti4, Elisée Wiita5, Ingrid Almlöf5, Olov Wallner5, Jonathan Davies4, Sara Košenina 4, Liuzhen Meng5, Maeve Long5, Oliver Mortusewicz 5, Geoffre...
7Z5S
Crystal Structure of botulinum neurotoxin A2 cell binding domain in complex with GD1a
Citation: Gregory, K.S.; Mahadeva, T.B.; Liu, S.M.; Acharya, K.R. Structural Features of Clostridium botulinum Neurotoxin Subtype A2 Cell Binding Domain. Toxins 2022, 14, 356. https://doi.org/10.3390/ toxins14050356 Received: 2 May 2022 Accepted: 18 May 2022 Published: 19 May 2022 Publisher’s Note: MDPI stays neutral w...
7Z5T
Crystal Structure of botulinum neurotoxin A2 cell binding domain
Citation: Gregory, K.S.; Mahadeva, T.B.; Liu, S.M.; Acharya, K.R. Structural Features of Clostridium botulinum Neurotoxin Subtype A2 Cell Binding Domain. Toxins 2022, 14, 356. https://doi.org/10.3390/ toxins14050356 Received: 2 May 2022 Accepted: 18 May 2022 Published: 19 May 2022 Publisher’s Note: MDPI stays neutral w...
7Z5U
Crystal structure of the peptidase domain of collagenase G from Clostridium histolyticum in complex with a hydroxamate-based inhibitor
Discovery and Characterization of Synthesized and FDA-Approved Inhibitors of Clostridial and Bacillary Collagenases Alaa Alhayek,⊥Ahmed S. Abdelsamie,⊥Esther Schönauer, Virgyl Camberlein, Evelyn Hutterer, Gernot Posselt, Jamil Serwanja, Constantin Blöchl, Christian G. Huber, Jörg Haupenthal, Hans Brandstetter, Silja We...
7Z5Y
CRYSTAL STRUCTURE OF WEISSELLA VIRIDESCENS FEMXVV NON-RIBOSOMAL AMINO ACID TRANSFERASE IN COMPLEX WITH A PEPTIDYL-XNA CONJUGATE
Published online 9 November 2022 Nucleic Acids Research, 2022, Vol. 50, No. 20 11415–11425 https://doi.org/10.1093/nar/gkac1023 Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis Lauriane Rietmeyer 1,†, In`es Li De La Sierra-Gallay 2,†, Guy Schepers3, Delphine Dorchˆene1, Laura Iannazzo4, Delphine ...
7Z5Z
CRYSTAL STRUCTURE OF WEISSELLA VIRIDESCENS FEMXVV NON-RIBOSOMAL AMINO ACID TRANSFERASE IN COMPLEX WITH A PEPTIDYL-XNA CONJUGATE
Published online 9 November 2022 Nucleic Acids Research, 2022, Vol. 50, No. 20 11415–11425 https://doi.org/10.1093/nar/gkac1023 Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis Lauriane Rietmeyer 1,†, In`es Li De La Sierra-Gallay 2,†, Guy Schepers3, Delphine Dorchˆene1, Laura Iannazzo4, Delphine ...
7Z61
Crystal structure of PI3Kgamma with a dihydropurinone inhibitor (compound 18)
Optimization of hERG and Pharmacokinetic Properties for Basic Dihydro‑8H‑purin-8-one Inhibitors of DNA-PK Frederick W. Goldberg,* Attilla K. T. Ting, David Beattie, Gillian M. Lamont, Charlene Fallan, M. Raymond V. Finlay, Beth Williamson, Marianne Schimpl, Alexander R. Harmer, Oladipupo B. Adeyemi, Pär Nordell, Anna S...
7Z6A
CRYSTAL STRUCTURE OF WEISSELLA VIRIDESCENS FEMXVV NON-RIBOSOMAL AMINO ACID TRANSFERASE IN COMPLEX WITH A PEPTIDYL-XNA CONJUGATE
Published online 9 November 2022 Nucleic Acids Research, 2022, Vol. 50, No. 20 11415–11425 https://doi.org/10.1093/nar/gkac1023 Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis Lauriane Rietmeyer 1,†, In`es Li De La Sierra-Gallay 2,†, Guy Schepers3, Delphine Dorchˆene1, Laura Iannazzo4, Delphine ...
7Z6B
PET hydrolase PET6 from halophilic organsim Vibrio gazogenes
F U L L - L E N G T H P A P E R Investigation of the halophilic PET hydrolase PET6 from Vibrio gazogenes Sebastian Weigert1 | Pablo Perez-Garcia2 | Florian J. Gisdon1 | Andreas Gagsteiger1 | Kristine Schweinshaut1 | G. Matthias Ullmann3 | Jennifer Chow2 | Wolfgang R. Streit2 | Birte Höcker1 1Department of Biochemistry,...
7Z6C
Crystal structure of human Dihydroorotate Dehydrogenase in complex with the inhibitor 2-Hydroxy-N-(2-ispropyl-5-methyl-4-phenoxyphenyl)pyrazolo[1,5-a]pyridine-3-carboxamide.
Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2‑Hydroxypyrazolo[1,5‑a]pyridine Scaffold: SAR of the Aryloxyaryl Moiety Stefano Sainas,§§ Marta Giorgis,§§ Paola Circosta, Giulio Poli, Marta Alberti, Alice Passoni, Valentina Gaidano, Agnese C. Pippione, Nicol...
7Z6F
Crystal structure of the substrate-binding protein YejA in complex with peptide fragment
PNAS  2025  Vol. 122  No. 1 e2319483121 https://doi.org/10.1073/pnas.2319483121 1 of 10 RESEARCH ARTICLE |  Significance The need for antibiotics that target infections from gram- negative pathogens is a growing global health concern. Here, we show that antibiotics with activity against gram-positive organisms c...