inchikey
stringlengths
27
27
name
stringlengths
5
122
smiles
stringlengths
1
323
logka
float64
0
12
source
stringclasses
3 values
n_heavy
int64
1
91
scaffold_family
stringclasses
5 values
known_scaffold
bool
2 classes
tmax_known
float64
0
1
is_novel
bool
2 classes
AAIHWHGLVCKBGZ-UHFFFAOYSA-N
AAIHWHGLVCKBGZ
CC(C)C#CCNC=O
null
qm9
9
null
false
0.1026
true
AAIIOHLTLWEMCP-UHFFFAOYSA-N
AAIIOHLTLWEMCP
C1NC1C12OC3CC1C32
null
qm9
9
null
false
0.129
true
AAIIZTWLPBIJGA-CXUHLZMHSA-N
AAIIZTWLPBIJGA
Oc1ccccc1/C=N/NC(=S)NC1CC2C=CC1C2
null
geom_drugs
20
null
false
0.0897
true
AAIJCFQQRWBAFC-HEFXARFJSA-N
AAIJCFQQRWBAFC
CCn1c(SCC(=O)N/N=C/C=C\c2ccccc2[N+](=O)[O-])nc2ccccc21
null
geom_drugs
29
null
false
0.1209
true
AAIJEURQKZASKQ-UHFFFAOYSA-N
AAIJEURQKZASKQ
Cc1ccc(F)c(C)c1
null
qm9
9
null
false
0.1273
true
AAIKREZGUXVKTN-UHFFFAOYSA-N
AAIKREZGUXVKTN
COc1ccc(C(=O)CN2CCN(c3ccc(F)cc3)CC2)cc1
null
geom_drugs
24
null
false
0.1884
true
AAIKZASNSMAOGO-UHFFFAOYSA-N
AAIKZASNSMAOGO
c1cnccncoc1
null
qm9
9
null
false
0.0508
true
AAILEWXSEQLMNI-UHFFFAOYSA-N
AAILEWXSEQLMNI
O=c1cccn[nH]1
null
geom_drugs
7
null
false
0.1111
true
AAIMXWPKUBSQNM-UHFFFAOYSA-N
AAIMXWPKUBSQNM
Cc1oc(-c2ccccc2Cl)nc1CS(=O)CC(=O)NCc1ccco1
null
geom_drugs
26
null
false
0.1266
true
AAINVONCQMFNEO-UHFFFAOYSA-N
AAINVONCQMFNEO
CC(C#N)C1(O)CC1O
null
qm9
9
null
false
0.2143
true
AAINWHXBUKJDJF-UHFFFAOYSA-N
AAINWHXBUKJDJF
NS(=O)(=O)c1ccc(NC=C2C(=O)OC3(CCCCC3)OC2=O)cc1
null
geom_drugs
25
null
false
0.1034
true
AAIOPLKMESRUOC-UHFFFAOYSA-N
AAIOPLKMESRUOC
O=C(NC1CCCC1)c1ccc(CS(=O)(=O)Cc2ccccc2F)o1
null
geom_drugs
25
null
false
0.1408
true
AAIOXXIRNCHNMB-UHFFFAOYSA-N
AAIOXXIRNCHNMB
O=C(CC1C(=O)NCCN1C(=O)Nc1ccc(F)cc1F)Nc1ccc(F)cc1
null
geom_drugs
29
null
false
0.1184
true
AAISMRVATULTLV-UHFFFAOYSA-N
AAISMRVATULTLV
O=S(=O)(NCc1cccnc1)c1cc(Cl)ccc1Cl
null
geom_drugs
19
null
false
0.1111
true
AAISTUFXBZKBEU-UHFFFAOYSA-N
AAISTUFXBZKBEU
COCC1(CO)CCO1
null
qm9
9
null
false
0.2692
true
AAISUDVSXFOHOW-LFIBNONCSA-N
AAISUDVSXFOHOW
Cc1ccc2cc(/C=C(\C#N)C(N)=O)c(N3CCCCC3)nc2c1
null
geom_drugs
24
null
false
0.1818
true
AAITUNLWLVHUMS-RIYZIHGNSA-N
AAITUNLWLVHUMS
CC(=O)N/N=C/c1c(C)[nH]n(-c2ccccc2)c1=O
null
geom_drugs
19
null
false
0.1385
true
AAITYCASMPCAAB-UHFFFAOYSA-N
AAITYCASMPCAAB
O=CC(=O)N1CC2CC21
null
qm9
9
null
false
0.129
true
AAIUAISLYPTWHT-UHFFFAOYSA-N
AAIUAISLYPTWHT
CN1C2C3OC(C3O)C21
null
qm9
9
null
false
0.0714
true
AAIUCVHMISBIEU-UHFFFAOYSA-N
AAIUCVHMISBIEU
CC(=O)NCCn1ccc2ccccc21
null
geom_drugs
15
null
false
0.1754
true
AAIUSJQCOVGWTL-UHFFFAOYSA-N
AAIUSJQCOVGWTL
CC1CC(C#N)C2CN12
null
qm9
9
null
false
0.0976
true
AAIVVQDGLIMYBQ-RFPFOJJUSA-N
AAIVVQDGLIMYBQ
O=C(NN1C(=O)C2C3C=CC([C@@H]2C1=O)C31CC1)c1ccccc1
null
geom_drugs
23
null
false
0.129
true
AAIVVQDGLIMYBQ-UHFFFAOYSA-N
AAIVVQDGLIMYBQ
O=C(NN1C(=O)C2C(C1=O)C1C=CC2C12CC2)c1ccccc1
null
geom_drugs
23
null
false
0.129
true
AAIYARYQJOBWIE-VULFUBBASA-N
AAIYARYQJOBWIE
COc1cccc(C(=O)N/N=C/c2ccc(OC)c(COc3ccccc3C(N)=O)c2)c1
null
geom_drugs
32
null
false
0.125
true
AAIYDYZRMWSWKI-UHFFFAOYSA-N
AAIYDYZRMWSWKI
CC12NC1CC1(O)CC12
null
qm9
9
null
false
0.2143
true
AAIYJZKKBMDVSP-UHFFFAOYSA-N
AAIYJZKKBMDVSP
O=[N+]([O-])c1ccc(C2=Nc3cc(Cl)ccc3OC2)cc1
null
geom_drugs
20
null
false
0.1081
true
AAJDSJCBTBMOPG-UHFFFAOYSA-N
AAJDSJCBTBMOPG
CCCC12OC3C1CC32
null
qm9
9
null
false
0.2222
true
AAJGLQBFERJSSV-UHFFFAOYSA-N
AAJGLQBFERJSSV
CCn1c(CNC(=O)c2cccc(C)c2)nnc1SCC(=O)NC1CCCC1
null
geom_drugs
28
null
false
0.15
true
AAJGTVXRCUDTNQ-CIAFOILYSA-N
AAJGTVXRCUDTNQ
O=C(N/N=C/c1ccco1)c1cccc(NC(=O)c2ccccc2Cl)c1
null
geom_drugs
26
null
false
0.1067
true
AAJHBUBXFOFUFH-UHFFFAOYSA-N
AAJHBUBXFOFUFH
Nc1cnc(O)oc1=O
null
qm9
9
null
false
0.1167
true
AAJHNBNHSXRALI-UHFFFAOYSA-N
AAJHNBNHSXRALI
C#CC1(C#N)OC1C#N
null
qm9
9
null
false
0.0645
true
AAJHOEQMTSTUJP-UHFFFAOYSA-N
AAJHOEQMTSTUJP
CCN(Cc1ccccc1)C(=O)C1CCN(S(=O)(=O)c2ccc3c(c2)OCCO3)CC1
null
geom_drugs
31
null
false
0.1277
true
AAJINUUEBDIAGI-UHFFFAOYSA-N
1-(2-Cyanophenyl)-3-(4-fluorophenyl)thiourea
N#Cc1ccccc1NC(=S)Nc1ccc(F)cc1
null
geom_drugs
19
null
false
0.0909
true
AAJIOFUVLXKEJB-UHFFFAOYSA-N
AAJIOFUVLXKEJB
CC(=O)c1ccc(NC(=O)COC(=O)c2ccccc2Nc2ccccc2)cc1
null
geom_drugs
29
null
false
0.1667
true
AAJIXYYFUWHLKI-UHFFFAOYSA-N
AAJIXYYFUWHLKI
CCOc1ccc(NC(=O)CNC(=O)c2ccco2)cc1
null
geom_drugs
21
null
false
0.2063
true
AAJJHYDKLWTJCD-UHFFFAOYSA-N
AAJJHYDKLWTJCD
O=C(Cn1ncc2c1-c1ccccc1OC2)N1CCN(c2ccccn2)CC1
null
geom_drugs
28
null
false
0.1446
true
AAJJLMKTUZDHEC-UHFFFAOYSA-N
AAJJLMKTUZDHEC
CCN1CCN(C(=S)Nc2cccc(C(F)(F)F)c2)CC1
null
geom_drugs
21
null
false
0.1304
true
AAJKAKDFFNGTCX-UHFFFAOYSA-N
AAJKAKDFFNGTCX
COC1CNCC(=O)C1
null
qm9
9
null
false
0.1562
true
AAJLDCPLKAAORC-UHFFFAOYSA-N
AAJLDCPLKAAORC
CC12CCC(C=O)C1O2
null
qm9
9
null
false
0.122
true
AAJLRXQUJXOGTL-MTEHDHEFSA-N
AAJLRXQUJXOGTL
COc1ccccc1/C=C/C=N/NC(=O)c1cnccn1
null
geom_drugs
21
null
false
0.1013
true
AAJNCMAXGCXPSF-CPNJWEJPSA-N
AAJNCMAXGCXPSF
Clc1ccc(N2CCN(/N=C/c3ccncc3)CC2)cc1
null
geom_drugs
21
null
false
0.1846
true
AAJNTGYUCARMSA-UHFFFAOYSA-N
AAJNTGYUCARMSA
COCCn1nnnc1C1(N(Cc2cc3cc(C)ccc3[nH]c2=O)CC2CCCO2)CCN(C)CC1
null
geom_drugs
36
null
false
0.1569
true
AAJOPMHTWQOBSN-UHFFFAOYSA-N
AAJOPMHTWQOBSN
S=C(NCCc1ccccn1)Nc1ccc(Cl)c(Cl)c1
null
geom_drugs
20
null
false
0.1194
true
AAJPBGSVEDDJSI-UHFFFAOYSA-N
AAJPBGSVEDDJSI
CC(C)(C)NC(=O)C1Cc2ccccc2CN1S(=O)(=O)c1ccc(F)cc1
null
geom_drugs
27
null
false
0.1111
true
AAJPKRBDZASFOT-UHFFFAOYSA-N
AAJPKRBDZASFOT
CC(OC(=O)c1ccccc1NS(=O)(=O)c1cccc(N)c1)C(=O)N(C)Cc1ccccc1
null
geom_drugs
33
null
false
0.1688
true
AAJQTWWVKREOQP-UHFFFAOYSA-N
AAJQTWWVKREOQP
O=C(O)CCC(=O)c1ccc2ccc3cccc4ccc1c2c34
null
geom_drugs
23
null
false
0.1818
true
AAJRGFLICCXVHY-UHFFFAOYSA-N
AAJRGFLICCXVHY
CC1C2CC1(C)C2CO
null
qm9
9
null
false
0.1852
true
AAJSLLAMJKOTMI-UHFFFAOYSA-N
AAJSLLAMJKOTMI
O=C(CSc1ncn[nH]1)Nc1cc(S(=O)(=O)N2CCCC2)ccc1Cl
null
geom_drugs
25
null
false
0.1176
true
AAJSORZPWSFOMG-UHFFFAOYSA-N
AAJSORZPWSFOMG
CCOC(=O)C1CCN(C(=O)CN(c2ccc3c(c2)OCCO3)S(C)(=O)=O)CC1
null
geom_drugs
29
null
false
0.1395
true
AAJXZKMGUIMSEV-UHFFFAOYSA-N
AAJXZKMGUIMSEV
COc1ccc(C2CC(O)(c3ccccc3)Oc3cc(OC)ccc32)cc1
null
geom_drugs
27
null
false
0.1224
true
AAJZGIJQXHXUCX-UHFFFAOYSA-N
AAJZGIJQXHXUCX
Cc1ccccc1NC(=O)CN1CCN(Cc2ccccc2)CC1
null
geom_drugs
24
null
false
0.1803
true
AAKBJLBKEFORKA-UHFFFAOYSA-N
AAKBJLBKEFORKA
c1onc2c1CNC2
null
qm9
8
null
false
0.1228
true
AAKBKSANSMEPRC-UHFFFAOYSA-N
1H-indol-2-yl(morpholin-4-yl)methanone
O=C(c1cc2ccccc2[nH]1)N1CCOCC1
null
geom_drugs
17
null
false
0.2031
true
AAKDIVRPNMEHQS-UHFFFAOYSA-N
AAKDIVRPNMEHQS
CC(C)(C)c1cc(C(=O)NCC(=O)OCC(=O)c2cccc([N+](=O)[O-])c2)cc(C(C)(C)C)c1
null
geom_drugs
33
null
false
0.1528
true
AAKDMZQFSPTWBO-UHFFFAOYSA-N
AAKDMZQFSPTWBO
CC1CN(c2ccc(Cl)cc2)c2nc3c(c(=O)[nH]c(=O)n3C)n2C1
null
geom_drugs
24
null
false
0.1867
true
AAKDPCMOSKMCJP-UHFFFAOYSA-N
AAKDPCMOSKMCJP
COC(=O)CCN1CCN(S(=O)(=O)c2cccc(Br)c2)CC1
null
geom_drugs
22
null
false
0.1467
true
AAKGITIJYOFIBH-UHFFFAOYSA-N
AAKGITIJYOFIBH
O=C(NCc1cccs1)C1CC(c2ccc(Cl)c(Cl)c2)=NO1
null
geom_drugs
22
null
false
0.1235
true
AAKIMHLJHRBNET-UHFFFAOYSA-N
AAKIMHLJHRBNET
CC1CN(c2ccc([N+](=O)[O-])c(N3CCCCC3)c2)CCN1
null
geom_drugs
22
null
false
0.1806
true
AAKIVSYPQBEFNF-ZPHPHTNESA-N
AAKIVSYPQBEFNF
COc1ccc(/C(O)=C2/C(=O)C(=O)N(c3ncccn3)C2c2ccc(F)cc2)cc1
null
geom_drugs
30
null
false
0.1071
true
AAKJBOXANFFSDJ-UHFFFAOYSA-N
AAKJBOXANFFSDJ
CCC1C2C(=O)C3C2N13
null
qm9
9
null
false
0.1613
true
AAKJLRGGTJKAMG-UHFFFAOYSA-O
AAKJLRGGTJKAMG
C#Cc1cccc([NH2+]c2ncnc3cc(OCCOC)c(OCCOC)cc23)c1
null
geom_drugs
29
null
false
0.0926
true
AAKKTZPXZJLQRE-UHFFFAOYSA-N
AAKKTZPXZJLQRE
COc1ccc(C(=O)N2CCN(C(=O)C3COc4ccccc4O3)CC2)cc1
null
geom_drugs
28
null
false
0.1013
true
AAKMJXBIIHGEFU-UHFFFAOYSA-N
AAKMJXBIIHGEFU
CCOC(=O)N1CCC(NC(=O)C2CCN(S(=O)(=O)N3CCC(C)CC3)CC2)CC1
null
geom_drugs
30
null
false
0.0833
true
AAKNZVGEPPGBGK-UHFFFAOYSA-N
AAKNZVGEPPGBGK
C#CC1(C)OC1C#N
null
qm9
8
null
false
0.0769
true
AAKOAFHGLFVXOR-UHFFFAOYSA-N
AAKOAFHGLFVXOR
CCOC(=O)CN(c1ccccn1)S(=O)(=O)c1ccc(OC)cc1
null
geom_drugs
24
null
false
0.1264
true
AAKOJKQMPSAJIG-UHFFFAOYSA-N
AAKOJKQMPSAJIG
COc1ccc(OC)c(NC(=O)Nc2cccc(Cn3cccn3)c2)c1
null
geom_drugs
26
null
false
0.1467
true
AAKOYCVQAYQRIG-JFLMPSFJSA-N
AAKOYCVQAYQRIG
O=C(O)c1ccc(/C=N/NC(=O)c2ccc(CN3c4cccc5cccc(c45)S3(=O)=O)cc2)cc1
null
geom_drugs
35
null
false
0.16
true
AAKQZDCEBUKFHD-UHFFFAOYSA-N
3-(4-chlorophenyl)-5-(1,1,2,2-tetrafluoroethyl)-1H-pyrazole
FC(F)C(F)(F)c1cc(-c2ccc(Cl)cc2)n[nH]1
null
geom_drugs
18
null
false
0.1194
true
AAKSJEDIWKZHQD-UHFFFAOYSA-N
AAKSJEDIWKZHQD
CCOC(=O)C1(CCCc2ccccc2)CCN(C(=O)c2cnn(CC)c2)CC1
null
geom_drugs
29
null
false
0.1149
true
AAKSNWHRVQHZEW-UHFFFAOYSA-N
AAKSNWHRVQHZEW
COc1cc(CN2CCCC(C(=O)Nc3ccccc3Oc3cccnc3)C2)ccc1F
null
geom_drugs
32
null
false
0.1222
true
AAKSTVXHRNNNGZ-UHFFFAOYSA-N
AAKSTVXHRNNNGZ
Clc1ccc(-n2nnnc2CN2CCOCC2)cc1
null
geom_drugs
19
null
false
0.1449
true
AAKUGLDBNILBQK-UHFFFAOYSA-N
AAKUGLDBNILBQK
COc1ccc(N2C(=O)CSC2c2cccc(OC)c2OC)cc1
null
geom_drugs
24
null
false
0.1039
true
AAKUOVDEBIZSJE-UHFFFAOYSA-N
AAKUOVDEBIZSJE
O=C(CN1C(=O)c2ccccc2C1=O)Nc1cccnc1
null
geom_drugs
21
null
false
0.1452
true
AAKUPJTYLNKERK-ACAGNQJTSA-N
AAKUPJTYLNKERK
CC1C(=O)NN=C1C(=O)N/N=C\c1ccc(O)cc1O
null
geom_drugs
20
null
false
0.1757
true
AAKVSQKPLNUJKV-UHFFFAOYSA-N
AAKVSQKPLNUJKV
C#CC1OCC(C)C1=O
null
qm9
9
null
false
0.1935
true
AAKWMGDOOVHENN-UHFFFAOYSA-N
AAKWMGDOOVHENN
CCOc1ccc(C2c3[nH]c4ccccc4c3CCN2CCCn2cccn2)cc1
null
geom_drugs
30
null
false
0.1364
true
AAKYALYUIAIXEB-UHFFFAOYSA-N
AAKYALYUIAIXEB
Cc1ccc(CCN2C(=O)CCC2(C)C(=O)NCc2cccnc2)cc1
null
geom_drugs
26
null
false
0.1467
true
AAKZCIHQRMMMAC-UHFFFAOYSA-N
AAKZCIHQRMMMAC
CCOC(=O)CCCCC(=O)c1[nH]c(=O)[nH]c1CSc1nnc2c3cc(Br)ccc3n(C)c2n1
null
geom_drugs
34
null
false
0.134
true
AALAMDHRAXQYQW-UHFFFAOYSA-N
AALAMDHRAXQYQW
CC(OC(=O)c1ccco1)C(=O)NC1CCCCC1
null
geom_drugs
19
null
false
0.1538
true
AALBSNQDJDYHSI-UHFFFAOYSA-N
AALBSNQDJDYHSI
O=C(NCC(c1cccs1)N1CCOCC1)c1ccccc1NS(=O)(=O)c1ccc(Br)cc1
null
geom_drugs
33
null
false
0.1209
true
AALBWBPELQNTGL-UHFFFAOYSA-N
AALBWBPELQNTGL
CCN(C(=O)COC(=O)c1cccn1C)C1CCS(=O)(=O)C1
null
geom_drugs
22
null
false
0.1098
true
AALCHAKPJXCSQC-UHFFFAOYSA-N
AALCHAKPJXCSQC
O=C(NCCc1ccccc1)c1ccccc1NC(=O)C1CCCCC1C(=O)O
null
geom_drugs
29
null
false
0.1642
true
AALFHFWRWXELGR-UHFFFAOYSA-N
AALFHFWRWXELGR
O=C(CSc1nc2ccccc2[nH]1)Nc1ccccc1N1CCOCC1
null
geom_drugs
26
null
false
0.2237
true
AALFXMWXGAJNMT-UHFFFAOYSA-N
AALFXMWXGAJNMT
CC1C2COC2C2OC12
null
qm9
9
null
false
0.0769
true
AALHCMPYVOKBEC-UHFFFAOYSA-N
AALHCMPYVOKBEC
CC12CC(N)C1(C#N)O2
null
qm9
9
null
false
0.1613
true
AALHEJVFGKQASC-UHFFFAOYSA-N
AALHEJVFGKQASC
CCOc1ccccc1OCC(=O)Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1
null
geom_drugs
30
null
false
0.1286
true
AALHTVFNLNVHJX-UHFFFAOYSA-N
AALHTVFNLNVHJX
Cc1nc(-c2cn[nH]c2-c2ccc(O)cc2O)cs1
null
geom_drugs
19
null
false
0.1739
true
AALICEQLWZCSCB-UHFFFAOYSA-N
AALICEQLWZCSCB
C#CC(C#N)CC(C)O
null
qm9
9
null
false
0.0682
true
AALIMZKVFUIMTO-UHFFFAOYSA-N
AALIMZKVFUIMTO
COCCCNc1oc(-c2ccccc2F)nc1C#N
null
geom_drugs
20
null
false
0.1392
true
AALJBWFAPIPTGL-UHFFFAOYSA-N
AALJBWFAPIPTGL
O=C1C=CC2(CO2)C1O
null
qm9
9
null
false
0.1579
true
AALJDLQELQAHIE-UHFFFAOYSA-N
AALJDLQELQAHIE
CCOC(=O)c1[nH]c(=O)[nH]c1CSc1ccccn1
null
geom_drugs
19
null
false
0.1311
true
AALJFFRFEBGHPM-UHFFFAOYSA-N
AALJFFRFEBGHPM
CC(C)OC(=O)CNc1n[nH]c(=S)[nH]c1=O
null
geom_drugs
16
null
false
0.127
true
AALKGALVYCZETF-UHFFFAOYSA-N
AALKGALVYCZETF
CCC(O)C(O)CO
null
qm9
8
null
false
0.1364
true
AALMRCUSSDYMBE-UHFFFAOYSA-N
AALMRCUSSDYMBE
COc1ccc(C2C=C(C)Nc3nc4ccccc4n32)cc1
null
geom_drugs
22
null
false
0.12
true
AALOEZGCFHDEHM-UHFFFAOYSA-N
AALOEZGCFHDEHM
N#Cc1c(N)n[nH]c1CCCN
null
geom_drugs
12
null
false
0.2
true
AALOKJJBOZKMIL-UHFFFAOYSA-N
AALOKJJBOZKMIL
CC1=C(C#N)C(=O)NC1
null
qm9
9
null
false
0.125
true
AALPCSZCRJQTNT-UHFFFAOYSA-N
AALPCSZCRJQTNT
C#CCn1nnc(C)n1
null
qm9
9
null
false
0.082
true
AALPWUGBAOXTOC-UHFFFAOYSA-N
AALPWUGBAOXTOC
CCN(CC)CCCNC(=O)CCC(=O)NNc1nc2ccccc2c2nc(C)nn12
null
geom_drugs
31
null
false
0.1375
true
AALQRZYXRYPZSN-UHFFFAOYSA-N
AALQRZYXRYPZSN
Cc1ccc(O)c(C(=O)CC(=O)c2ccc(Cl)cc2)c1
null
geom_drugs
20
null
false
0.1333
true
AALQZTJWQWHSPB-UHFFFAOYSA-N
AALQZTJWQWHSPB
COCCCN(C(C)=O)c1nc(-c2ccc(OC)cc2)cs1
null
geom_drugs
22
null
false
0.1154
true